Bulletin of the Korean Chemical Society

Korean Chemical Society (대한화학회)
권호 표지
DOI QR코드

DOI QR Code

Discovery of 2-Aminothiazole Derivatives as Antitumor Agents

  • Li, Minghua (Department of Chemistry, College of Natural Science, Chung-Ang University) ;
  • Sim, Yoo-Jin (Department of Chemistry, College of Natural Science, Chung-Ang University) ;
  • Ham, Seung-Wook (Department of Chemistry, College of Natural Science, Chung-Ang University)
  • Received : 2010.03.02
  • Accepted : 2010.04.05
  • Published : 2010.06.20
Download PDF
⟨ Previous Next ⟩

Abstract

Keywords

References

  1. Conrath, U.; Pieterse, C. M.; Mauch-Mani, B. Trends. Plant Sci. 2002, 7, 210. https://doi.org/10.1016/S1360-1385(02)02244-6
  2. Kim, K. S.; Kimball, S. D.; Misra, R. N.; Rawlins, D. B.; Hunt, J. T.; Xiao, H. Y.; Lu, S.; Qian, L.; Han, W. C.; Shan, W.; Mitt, T.; Cai, Z. W.; Poss, M. A.; Zhu, H.; Sack, J. S.; Tokarski, J. S.; Chang, C. Y.; Pavletich, N.; Kamath, A.; Humphreys, W. G.; Marathe, P.; Bursuker, I.; Kellar, K. A.; Roongta, U.; Batorsky, R.; Mulheron, J. G.; Bol, D.; Fairchild, C. R.; Lee, F. Y.; Webster, K. R. J. Med. Chem. 2002, 45, 3905. https://doi.org/10.1021/jm0201520
  3. Misra, R. N.; Xiao, H. Y.; Kim, K. S.; Lu, S.; Han, W. C.; Barbosa, S. A.; Hunt, J. T.; Rawlins, D. B.; Shan, W.; Ahmed, S. Z.; Qian, L.; Chen, B. C.; Zhao, R.; Bednarz, M. S.; Kellar, K. A.; Mulheron, J. G.; Batorsky, R.; Roongta, U.; Kamath, A.; Marathe, P.; Ranadive, S. A.; Sack, J. S.; Tokarski, J. S.; Pavletich, N. P.; Lee, F. Y.; Webster, K. R.; Kimball, S. D. J. Med. Chem. 2004, 47, 1719. https://doi.org/10.1021/jm0305568
  4. Borzilleri, R. M.; Bhide, R. S.; Barrish, J. C.; D'Arienzo, C. J.; Derbin, G. M.; Fargnoli, J.; Hunt, J. T.; Jeyaseelan, R. Sr.; Kamath, A.; Kukral, D. W.; Marathe, P.; Mortillo, S.; Qian, L.; Tokarski, J. S.; Wautlet, B. S.; Zheng, X.; Lombardo, L. J. J. Med. Chem. 2006, 49, 3766. https://doi.org/10.1021/jm060347y
  5. Helal, C. J.; Sanner, M. A.; Cooper, C. B.; Gant, T.; Adam, M.; Lucas, J. C.; Kang, Z.; Kupchinsky, S. Ahlijanian, M. K.; Tate, B.; Menniti, F. S.; Kelly, K.; Peterson, M. Bioorg. Med. Chem. Lett. 2004, 14, 5521. https://doi.org/10.1016/j.bmcl.2004.09.006
  6. Halland, N.; Braunton, A.; Bachmann, S.; Marigo, M.; Jorgensen, K. A. J. Am. Chem. Soc. 2004, 126, 4790. https://doi.org/10.1021/ja049231m
  7. Minko, T.; Kopeckova, P.; Pozharov, V.; Kopecek, J. J. Controlled Release 1998, 54, 223. https://doi.org/10.1016/S0168-3659(98)00009-1
  8. Williams, G. T. Cell 1991, 65, 1097. https://doi.org/10.1016/0092-8674(91)90002-G

Cited by

  1. Synthesis and antitumor activity of 4-tert-butyl-5-benzyl-2-benzyliminothiazoles vol.30, pp.1, 2014, https://doi.org/10.1007/s40242-013-3345-6
  2. @KSF and Evaluating Their Antibacterial and Antioxidant Activities vol.348, pp.4, 2015, https://doi.org/10.1002/ardp.201400414
  3. A novel schiff base ligand and its Ni(II) complex: synthesis and characterization vol.147, pp.12, 2016, https://doi.org/10.1007/s00706-016-1727-5
  4. Facile synthesis and biological assays of novel 2,4-disubstituted hydrazinyl-thiazoles analogs vol.20, pp.2, 2016, https://doi.org/10.1007/s11030-015-9654-7
  5. Efficient construction of C–N and C–S bonds in 2-iminothiazoles via cascade reaction of enaminones with potassium thiocyanate vol.15, pp.17, 2017, https://doi.org/10.1039/C7OB00306D
  6. )-dione derivatives vol.192, pp.10, 2017, https://doi.org/10.1080/10426507.2017.1354209
  7. A Novel Aminothiazole Derivative Induces Apoptosis and Cell Cycle Arrest in Tumor Cells vol.31, pp.11, 2010, https://doi.org/10.5012/bkcs.2010.31.11.3454
  8. 2-Aminothiazole Derivative as a New Class of TrkA Kinase Inhibitor vol.32, pp.8, 2011, https://doi.org/10.5012/bkcs.2011.32.8.2893
  9. Facile One-Pot Procedure for the Synthesis of 2-Aminothiazole Derivatives vol.85, pp.8, 2010, https://doi.org/10.3987/com-12-12510
  10. Identification of robust synthon in the molecular salts of 2-aminothiazole with substituted benzoic acids: A case study vol.126, pp.5, 2014, https://doi.org/10.1007/s12039-014-0693-x
  11. Synthesis and Bio-Evaluation of Novel N-(4-(8-Methoxy-2-Oxo-2H-Chromen-3-Yl) Thiazol-2-Yl) Amide Derivatives vol.71, pp.None, 2016, https://doi.org/10.18052/www.scipress.com/ilcpa.71.19
  12. Synthesis of Terminal Thiazoles from N-Protected Amino Acids and a Study of Their Antibacterial Activities vol.52, pp.3, 2010, https://doi.org/10.1080/00304948.2020.1721959
  13. Synthesis, Characterization and Bioassay of Novel Substituted 1-(3-(1,3-Thiazol-2-yl)phenyl)-5-oxopyrrolidines vol.25, pp.10, 2020, https://doi.org/10.3390/molecules25102433